Novel Pharmacology Approaches to GPCR Allosteric Modulation

Time: 2:00 pm
day: Pre Conference Focus Day

Details:

• Allosteric modulation of GPCRs is a promising approach for drug discovery
• The structural biology revolution has illuminated the basis for GPCR allosteric modulation by small molecules
• Describe the pharmacological and structural mechanisms of novel Class B GPCR allosteric modulators
• Discuss if current pharmacology models are sufficient to describe GPCR allosteric modulation