Novel Pharmacology Approaches to GPCR Allosteric Modulation

Time: 2:00 pm
day: Pre Conference Focus Day


  • Allosteric modulation of GPCRs is a promising approach for drug discovery
  • The structural biology revolution has illuminated the basis for GPCR allosteric modulation by small molecules
  • Describe the pharmacological and structural mechanisms of novel Class B GPCR allosteric modulators
  • Discuss if current pharmacology models are sufficient to describe GPCR allosteric modulation